Construct · 1 fields · 1 citations

covalent inhibitor: a standalone construct

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Medicinal chemistry

drug that forms a covalent bond with its target, often a cysteine, after first binding noncovalently, giving prolonged and potent inhibition.

In medicinal chemistry, covalent inhibitor refers to drug that forms a covalent bond with its target, often a cysteine, after first binding noncovalently, giving prolonged and potent inhibition. This meaning comes from Singh (2011) in Nature Reviews Drug Discovery.[1]

Unit
Recovery means
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Nearby constructs

binding4 fields · 4 citationsjingle · one word, four constructs bond2 fields · 2 citationsjingle · one word, two constructs inhibition4 fields · 4 citationsjingle · one word, four suppressions

References

Singh, J., Petter, R. C., Baillie, T. A., & Whitty, A. (2011). The resurgence of covalent drugs. Nature Reviews Drug Discovery, 10(4), 307-317. https://doi.org/10.1038/nrd3410

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